SL-01, p53/mdm2 inhibitor

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Product price

128 EUR

Product size

50 mg

Product catalog no.

SIH-343-50MG

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Additional description

Tissue, pathway, proteinase, peptidase, protease ,acrosin, lipoprotein, activator, caspase, trypsin, papain, esterase inhibitors are proteins or receptor ligands or receptor antagonists that bind to an enzyme receptor and decreases its activity. Since blocking an enzyme's activity can kill a pathogen or correct a metabolic imbalance, many drugs are enzyme inhibitors. Not all receptor antagonist that bind to enzymes are inhibitors; enzyme activator ligands or agonists bind to enzymes and increase their enzymatic activity, while enzyme substrates bind and are converted to products in the normal catalytic cycle of the enzyme.

Representative figure legend

Chemical structure of SL-01 (SIH-343), a p53/mdm2 inhibitor. CAS #: 26049-94-5. Molecular Formula: C18H18ClNO3. Molecular Weight: 331.8 g/mol. Chemical structure of SL-01, a p53/mdm2 inhibitor (SIH-343). CAS # 26049-94-5. Molecular Formula: C18H18ClNO3.

 

Safety information

Classification: Caution – Substance not yet fully tested. Safety Phrases: S22 - Do not breathe dust S36/37/39 - Wear suitable protective clothing, gloves and eye/face protection S24/25- Avoid contact with skin and eyes

Other name

Benzyl [(2S)-4-chloro-3-oxo-1-phenyl-2-butanyl]carbamate; N-Benzyloxycarbonyl-Lphenylalaninylchloromethyl ketone; ZPCK

 

Scientific context

Inhibits the p53-MDM2 interaction (20 µM). Has also been shown to inhibit bovine chymotrypsin A-y.

Primary research fields

Cancer, Apoptosis, Cancer Growth Inhibitors, p53/mdm2 Inhibitors

 

Soluble in

Soluble in 50 mg/ml DMSO oir 15 mg/ml warm Ethanol

Bibliography

1. Li J., et al. (2011) J Biol Screening 16: 450.

 

Purity pourcentage

>98% (TLC); NMR (Conforms)

Description

p53/mdm2 inhibitor

 

PubMed number

Refer to PubMed

Shipping recommendations

Shipped Ambient

 

Product category

Small Molecules

Warning information

Non-hazardous

 

Tested reactivity

To be tested

Tested applications

To be tested

 

Release date

17-Aug-2012

Molecular weight

331,8 g/mol

 

Physical appearance

White Solid

Chemical formula

C18H18ClNO3

 

CAS number

26049-94-5

Product type

Inhibitor

 

Origin

Synthetic

Stock availabilitIn Stock

In Stock

 

Storage recommendations

-20ºC

Country of production

Canada

 

PubChem number

99625

Total weight (kg)

0.25

 

Net weight (g)

0.05